| 產品名稱 | PH 797804 |
| 產品貨號 | Axon 1837 CAS [586379-66-0] MF C22H19BrF2N2O3MW 477.30 Purity: 99% Soluble in DMSO and ethanol Description Highly potent, selective and metabolically stable inhibitor of p38 MAPK (p38α cascade IC50: 2.3 nM); an ATP-competitive, readily reversible inhibitor of the α isoform of human p38 MAP kinase, exhibiting a Ki of 5.8 nM; clinical candidate. *PH 797804 is an (-)-atropisomer, which is 100-fold more potent than its (+)-atropisomer. Be careful that racemate of PH 797804 is wrongly provided by other supplier as drug PH 797804 itself. The less potent (+)-rotating atropisomer is also available (inquire). Be right about your drug. The racemate,?(±)-PH797804 (Axon 2786) is also available. |
| 產品價格 | 現貨詢價，電話：010-67529703 |
| 產品規格 | |
| 產品品牌 | axonmedchem |
| 產品概述 | |
| 產品詳情 |
PH 797804Axon 1837 CAS [586379-66-0] MF C22H19BrF2N2O3
DescriptionHighly potent, selective and metabolically stable inhibitor of p38 MAPK (p38α cascade IC50: 2.3 nM); an ATP-competitive, readily reversible inhibitor of the α isoform of human p38 MAP kinase, exhibiting a Ki of 5.8 nM; clinical candidate. *PH 797804 is an (-)-atropisomer, which is 100-fold more potent than its (+)-atropisomer. Be careful that racemate of PH 797804 is wrongly provided by other supplier as drug PH 797804 itself. The less potent (+)-rotating atropisomer is also available (inquire). Be right about your drug. The racemate,?(±)-PH797804 (Axon 2786) is also available. KEYWORDS: PH 797804 | supplier | p38 MAPK inhibitor | PH797804 | CAS [586379-66-0] | MAPK | MAPK (p38) | Inhibitor | Enzymes
Inhibitor of p38α MAPK
Chemical name3-(3-bromo-4-(2,4-difluorobenzyloxy)-6-methyl-2-oxopyridin-1(2H)-yl)-N,4-dimethylbenzamide Parent CAS No.[586379-66-0] |
| 產品資料 |
